Molecule Details
InChIKeyNKRSLISCOPHPJT-UHFFFAOYSA-N
Compound Name4-[[1-(4,4-Dimethylcyclohexyl)pyrazolo[3,4-d]pyrimidin-6-yl]amino]-1-methylpyrrole-2-carboxamide
Canonical SMILESCn1cc(Nc2ncc3cnn(C4CCC(C)(C)CC4)c3n2)cc1C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB