Molecule Details
InChIKeyNKORVPQBJCGYEC-UHFFFAOYSA-N
Compound NameDB-02197
Canonical SMILESNS(=O)(=O)c1ccc(Nc2nccc(-c3cnc4ccccn34)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.0
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB02197
Drug Name4-[(4-Imidazo[1,2-a]Pyridin-3-Ylpyrimidin-2-Yl)Amino]Benzenesulfonamide
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 7657 CHEMBL73303 ChemSpider: 4450680 PDB: HDT PubChem:5288527 PubChem:46504935 ZINC: ZINC000001493866
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06729 CD2 Homo sapiens Human PF05790 PF07686 9.0 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 9.0 pIC50 TTD_MultiTarget
DrugBank Target Actions (1)
Target Gene Target Name Action Type
P24941 CDK2 Cyclin-dependent kinase 2 binder targets