Molecule Details
InChIKeyNJMHKVAICPWFEV-UHFFFAOYSA-N
Compound Name1,1-Dioxo-2-[5-(4-pyridin-2-ylpiperazin-1-yl)pentyl]-1,2-benzothiazol-3-one
Canonical SMILESO=C1c2ccccc2S(=O)(=O)N1CCCCCN1CCN(c2ccccn2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P34969 HTR7 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB