Molecule Details
InChIKeyNJLNPETVWRAQNN-UHFFFAOYSA-N
Compound Name5,6-dimethyl-3-[3-[4-[2-(2,2,2-trifluoroethoxy)phenyl]piperazin-1-yl]propyl]-1H-pyrimidine-2,4-dione
Canonical SMILESCc1[nH]c(=O)n(CCCN2CCN(c3ccccc3OCC(F)(F)F)CC2)c(=O)c1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 10.4 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB