Molecule Details
InChIKeyNJCWASKCTHVLLT-UHFFFAOYSA-N
Compound Name6-Chloro-5-tert-butyl-1-(3-pyridylcarbamoyl)indoline
Canonical SMILESCC(C)(C)c1cc2c(cc1Cl)N(C(=O)Nc1cccnc1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB