Molecule Details
InChIKeyNIPJQRGYPGKSQY-UHFFFAOYSA-N
Compound Name3-N-[4-(3-morpholin-4-ylpropoxy)phenyl]-1-pyridin-2-yl-1,2,4-triazole-3,5-diamine
Canonical SMILESNc1nc(Nc2ccc(OCCCN3CCOCC3)cc2)nn1-c1ccccn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.92
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 7.9 Ki ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 7.9 pIC50 TTD_MultiTarget