Molecule Details
InChIKeyNIKCYGIZNVHYMC-HXUWFJFHSA-N
Compound Name9-fluoro-10-[(3R)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-ynyl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide
Canonical SMILESCc1cc([C@](C)(O)C#Cc2cc3c(cc2F)OCCn2cc(C(N)=O)nc2-3)no1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99558 MAP3K14 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
O00329 PIK3CD Homo sapiens Human PF00454 PF00792 PF02192 PF00794 PF00613 7.3 Ki ChEMBL
P27986 PIK3R1 Homo sapiens Human PF16454 PF00620 PF00017 7.3 Ki ChEMBL;BindingDB