Molecule Details
InChIKeyNHSDXYBXQGQSRA-UHFFFAOYSA-N
Compound NameN-cyclopentyl-4-(3-(tetrahydro-2H-pyran-3-yl)-1H-pyrazol-4-yl)pyrimidin-2-amine
Canonical SMILESc1cc(-c2c[nH]nc2C2CCCOC2)nc(NC2CCCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.9 Ki ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.6 IC50 ChEMBL
P53779 MAPK10 Homo sapiens Human PF00069 6.6 IC50 ChEMBL