Molecule Details
InChIKeyNHLHTGDNMWUOMW-UHFFFAOYSA-N
Compound Name5-[4-[4-(8-hydroxy-2-oxo-1H-quinolin-5-yl)piperazin-1-yl]butoxy]pyrazolo[1,5-a]pyridine-3-carbaldehyde
Canonical SMILESO=Cc1cnn2ccc(OCCCCN3CCN(c4ccc(O)c5[nH]c(=O)ccc45)CC3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB