Molecule Details
InChIKeyNGASNWUKBBDWEM-UHFFFAOYSA-N
Compound Name2-{4-[2-methyl-4-(quinolin-2-yl)piperazin-1-yl]butyl}-2,3-dihydro-1H-isoindole-1,3-dione
Canonical SMILESCC1CN(c2ccc3ccccc3n2)CCN1CCCCN1C(=O)c2ccccc2C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.99
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.1 IC50 ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB