Molecule Details
InChIKeyNFUKLMJHYQPDNT-UHFFFAOYSA-N
Compound Name8-(2-Methyl-1-oxidopyridin-1-ium-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
Canonical SMILESCc1c(Oc2sc(C(N)=O)c3c2-c2sncc2CC3)ccc[n+]1[O-]
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 8.4 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 8.4 IC50 ChEMBL
Q9BWU1 CDK19 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB