Molecule Details
InChIKeyNETRMZMGTHLSBM-ZDUSSCGKSA-N
Compound Name2-[4-[3-[(1S)-1-quinolin-6-ylethyl]triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol
Canonical SMILESC[C@@H](c1ccc2ncccc2c1)n1nnc2ncc(-c3cnn(CCO)c3)nc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08581 MET Homo sapiens Human PF07714 PF01437 PF01403 PF01833 8.9 IC50 ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 6.4 IC50 ChEMBL
Q14432 PDE3A Homo sapiens Human PF00233 6.2 IC50 ChEMBL