Molecule Details
InChIKeyNEOMSSISKDUIHW-PGCXCKJESA-N
Compound Name(2S)-2-acetamido-5-amino-N-[(2S)-2-[[(2S)-4-(diaminomethylideneamino)-2-[[1-[4-[1-[2-oxo-2-(6-oxo-5H-benzo[b][1,4]benzodiazepin-11-yl)ethyl]piperidin-4-yl]butyl]piperidin-4-yl]amino]butanoyl]amino]propanoyl]pentanamide
Canonical SMILESCC(=O)N[C@@H](CCCN)C(=O)NC(=O)[C@H](C)NC(=O)[C@H](CCNC(=N)N)NC1CCN(CCCCC2CCN(CC(=O)N3c4ccccc4NC(=O)c4ccccc43)CC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08172 CHRM2 Homo sapiens Human PF00001 9.8 Ki ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P08173 CHRM4 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB