Molecule Details
InChIKeyNEKNPPRWLZIEGE-UHFFFAOYSA-N
Compound Name5-[2-[4-[(2,5-Dichlorophenyl)methyl]piperazin-1-yl]ethoxy]-2-methylquinoline
Canonical SMILESCc1ccc2c(OCCN3CCN(Cc4cc(Cl)ccc4Cl)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB