Molecule Details
InChIKeyNEDWSVCVHMJKSZ-UHFFFAOYSA-N
Compound Name3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one
Canonical SMILESCOc1ccccc1N1CCN(CCCCN2CCc3cc(-c4ccco4)ccc3C2=O)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 8.5 Ki ChEMBL
P14416 DRD2 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB