Molecule Details
InChIKeyNDCWSHMFDBDIQV-UHFFFAOYSA-N
Compound NameN-((1H-imidazol-2-yl)methyl)-6-(benzo[d][1,3]dioxol-5-yl)-N-methylquinazolin-4-amine
Canonical SMILESCN(Cc1ncc[nH]1)c1ncnc2ccc(-c3ccc4c(c3)OCO4)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HAZ1 CLK4 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB
Q13627 DYRK1A Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB