Molecule Details
InChIKeyNDASMCYFWCEUSG-GFCCVEGCSA-N
Compound Name(R)-4-[3-(5-Chloro-pyrimidin-2-yloxy)-pyrrolidin-1-yl]-6,7-dimethoxy-quinazoline
Canonical SMILESCOc1cc2ncnc(N3CC[C@@H](Oc4ncc(Cl)cn4)C3)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 7.4 Ki ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 6.8 Ki ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 6.5 Ki ChEMBL;BindingDB