Molecule Details
InChIKeyNCSQDKMOKNQGSG-SFHVURJKSA-N
Compound Name(2s)-4-[2-Amino-6-(3-Amino-2h-Indazol-6-Yl)pyrimidin-4-Yl]-N-Phenylmorpholine-2-Carboxamide
Canonical SMILESNc1nc(-c2ccc3c(N)[nH]nc3c2)cc(N2CCO[C@H](C(=O)Nc3ccccc3)C2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 7.7 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 6.1 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 Clinical TTD_MultiTarget TTD_MultiTarget