Molecule Details
InChIKeyNCPSMBVBKJXJPP-UHFFFAOYSA-N
Compound Name4-[4-[2-(2H-tetrazol-5-yl)thieno[2,3-c]pyridin-4-yl]oxyphenyl]benzamide
Canonical SMILESNC(=O)c1ccc(-c2ccc(Oc3cncc4sc(-c5nn[nH]n5)cc34)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 8.5 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 8.5 IC50 ChEMBL
P41279 MAP3K8 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB