Molecule Details
InChIKeyNCJWLSWXMPGOIS-UHFFFAOYSA-N
Compound Name1-(1-{3-[1-Benzoyl-3-(3,4-dichloro-phenyl)-piperidin-3-yl]-propyl}-4-phenyl-piperidin-4-yl)-ethanone
Canonical SMILESCC(=O)C1(c2ccccc2)CCN(CCCC2(c3ccc(Cl)c(Cl)c3)CCCN(C(=O)c3ccccc3)C2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 8.8 IC50 ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 6.4 IC50 ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 6.3 IC50 ChEMBL;BindingDB