Molecule Details
InChIKeyNBMBJGUURXSJBY-UHFFFAOYSA-N
Compound NameN-(6-(1H-Imidazol-1-yl)pyridin-3-yl)-3-(cyclopropylmethyl)-7-methyl-3H-imidazo[4,5-b]pyridin-5-amine
Canonical SMILESCc1cc(Nc2ccc(-n3ccnc3)nc2)nc2c1ncn2CC1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18507 GABRG2 Homo sapiens Human PF02931 PF02932 7.8 Ki ChEMBL
P28472 GABRB3 Homo sapiens Human PF02931 PF02932 7.8 Ki ChEMBL
P31644 GABRA5 Homo sapiens Human PF02931 PF02932 7.8 Ki ChEMBL;BindingDB