Molecule Details
InChIKeyNBHYPBDUODSQHJ-DTPUHQDNSA-N
Compound NameVhl-IN-1
Canonical SMILESCc1cc(-c2scnc2C)ccc1[C@H](C)NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)C1(F)CC1)C(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.4
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15369 ELOC Homo sapiens Human PF03931 7.5 Kd ChEMBL
Q15370 ELOB Homo sapiens Human PF00240 7.5 Kd ChEMBL
P40337 VHL Homo sapiens Human PF01847 PF17211 7.2 IC50 ChEMBL