Molecule Details
InChIKeyNAUDEXJEXLGXTN-UHFFFAOYSA-N
Compound Name1-{2-[3-(4-Cyano-3-naphthalen-1-yl-benzyl)-3H-imidazol-4-yl]-acetyl}-5-methoxy-1,2,3,6-tetrahydro-pyridine-4-carbonitrile
Canonical SMILESCOC1=C(C#N)CCN(C(=O)Cc2cncn2Cc2ccc(C#N)c(-c3cccc4ccccc34)c2)C1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.85
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.8 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.8 IC50 ChEMBL