Molecule Details
InChIKeyNAHYDLCBWFSEJF-UHFFFAOYSA-N
Compound Name3-[4-(1-Phenylpyrazolo[5,4-d]pyrimidin-4-yl)piperazin-1-yl]benzonitrile
Canonical SMILESN#Cc1cccc(N2CCN(c3ncnc4c3cnn4-c3ccccc3)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11166 SLC2A1 Homo sapiens Human PF00083 7.4 IC50 ChEMBL;BindingDB
P11169 SLC2A3 Homo sapiens Human PF00083 7.2 IC50 ChEMBL;BindingDB
P11168 SLC2A2 Homo sapiens Human PF00083 6.7 IC50 ChEMBL;BindingDB