Molecule Details
InChIKeyMZUXZKDOYICLDH-SFYZADRCSA-N
Compound Name[(2S,5R)-2-[(6-amino-2-pyridinyl)carbamoyl]-7-oxo-1,6-diazabicyclo[3.2.1]octan-6-yl] hydrogen sulfate
Canonical SMILESNc1cccc(NC(=O)[C@@H]2CC[C@@H]3CN2C(=O)N3OS(=O)(=O)O)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.5
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q3LG62 ampC Pseudomonas aeruginosa Pathogen PF00144 8.1 IC50 BindingDB
I7AKP2 KPC-2 Klebsiella pneumoniae Pathogen PF13354 8.0 IC50 BindingDB
Q8RLA6 blaOXA-33 Acinetobacter baumannii Pathogen PF00905 6.4 IC50 ChEMBL;BindingDB