Molecule Details
InChIKeyMZRCCMMKNFJJEA-UHFFFAOYSA-N
Compound NameN-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}isonicotinamide
Canonical SMILESCc1cc(-c2nc3cccnn3c2-c2ccnc(NC(=O)c3ccncc3)c2)ccc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
O15264 MAPK13 Homo sapiens Human PF00069 7.8 IC50 ChEMBL
P53778 MAPK12 Homo sapiens Human PF00069 7.8 IC50 ChEMBL
Q15759 MAPK11 Homo sapiens Human PF00069 7.8 IC50 ChEMBL