Molecule Details
InChIKeyMZPQDMUNWXBKLC-UHFFFAOYSA-N
Compound Name2-acetyl-N-[5-[[2-(1-methylpyrazol-4-yl)-4-pyridinyl]oxy]-2-pyridinyl]-5-oxo-2,6-diazaspiro[3.4]octane-6-carboxamide
Canonical SMILESCC(=O)N1CC2(CCN(C(=O)Nc3ccc(Oc4ccnc(-c5cnn(C)c5)c4)cn3)C2=O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 8.7 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 8.3 IC50 ChEMBL;BindingDB
P16234 PDGFRA Homo sapiens Human PF07679 PF25305 PF07714 7.2 IC50 ChEMBL;BindingDB