Molecule Details
InChIKeyMZLGPWMELUQSRS-UHFFFAOYSA-N
Compound Name(5-(Aminomethyl)-2-(8-methoxy-2-(trifluoromethyl)quinolin-5-yl)oxazol-4-yl)(4-hydroxy-4-phenylpiperidin-1-yl)methanone
Canonical SMILESCOc1ccc(-c2nc(C(=O)N3CCC(O)(c4ccccc4)CC3)c(CN)o2)c2ccc(C(F)(F)F)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 8.7 IC50 ChEMBL;BindingDB
Q9HCR9 PDE11A Homo sapiens Human PF01590 PF00233 6.3 IC50 ChEMBL;BindingDB
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 6.2 IC50 ChEMBL;BindingDB