Molecule Details
InChIKeyMZEOWSVWCPCLAR-UHFFFAOYSA-N
Compound Name5-(4-(piperidin-1-yl)piperidin-1-yl)-2-(6-(trifluoromethyl)-1H-indazol-3-yl)-1H-benzo[d]imidazole
Canonical SMILESFC(F)(F)c1ccc2c(-c3nc4cc(N5CCC(N6CCCCC6)CC5)ccc4[nH]3)[nH]nc2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.7
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11362 FGFR1 Homo sapiens Human PF07679 PF00047 PF07714 8.7 pIC50 TTD_MultiTarget
P17948 FLT1 Homo sapiens Human PF07679 PF00047 PF13927 PF22971 PF07714 PF21339 PF17988 PF22854 8.7 IC50 ChEMBL;BindingDB