Molecule Details
InChIKeyMYPQPZOTEGVVQY-UHFFFAOYSA-N
Compound Name5-[3-Fluoro-4-({6-methoxy-7-[3-(morpholin-4-yl)propoxy]quinolin-4-yl}oxy)phenyl]-2-[(4-fluorophenyl)methyl]-3-methyl-3,4-dihydropyrimidin-4-one
Canonical SMILESCOc1cc2c(Oc3ccc(-c4cnc(Cc5ccc(F)cc5)n(C)c4=O)cc3F)ccnc2cc1OCCCN1CCOCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08581 MET Homo sapiens Human PF07714 PF01437 PF01403 PF01833 7.8 IC50 ChEMBL;BindingDB
P14210 HGF Homo sapiens Human PF00051 PF00024 PF00089 6.8 IC50 ChEMBL
Q04912 MST1R Homo sapiens Human PF07714 PF01437 PF01403 PF01833 6.2 Ki ChEMBL