Molecule Details
InChIKeyMYHOUKHXSVKHBA-UHFFFAOYSA-N
Compound Name4-[4-[3-[4-[(propan-2-ylamino)methyl]anilino]-1H-pyrazol-5-yl]phenyl]benzene-1,3-diol
Canonical SMILESCC(C)NCc1ccc(Nc2cc(-c3ccc(-c4ccc(O)cc4O)cc3)[nH]n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.99
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14757 CHEK1 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
O00141 SGK1 Homo sapiens Human PF00069 PF00433 6.5 IC50 ChEMBL;BindingDB
O96017 CHEK2 Homo sapiens Human PF00498 PF00069 Clinical TTD_MultiTarget TTD_MultiTarget