Molecule Details
InChIKeyMXRSDWOBSNRDKJ-ARJAWSKDSA-N
Compound Name4-amino-5-cyano-N-[(4-methylsulfonylphenyl)methyl]-6-[(Z)-prop-1-enyl]pyridine-2-carboxamide
Canonical SMILESC/C=C\c1nc(C(=O)NCc2ccc([S@SP2](C)(=O)=O)cc2)cc(N)c1C#N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB