Molecule Details
InChIKeyMXRHKEUIFABQMB-UHFFFAOYSA-N
Compound Name3-methyl-1-propan-2-yl-5-(2-propoxyphenyl)-N-(1H-pyrazol-4-ylmethyl)pyrazolo[4,5-b]pyridin-7-amine
Canonical SMILESCCCOc1ccccc1-c1cc(NCc2cn[nH]c2)c2c(n1)c(C)nn2C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.03
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 8.8 IC50 ChEMBL;BindingDB
P54750 PDE1A Homo sapiens Human PF00233 PF08499 7.7 IC50 ChEMBL;BindingDB
Q14123 PDE1C Homo sapiens Human PF00233 PF08499 7.6 IC50 ChEMBL;BindingDB