Molecule Details
InChIKeyMXFWWQICDIZSOA-UHFFFAOYSA-N
Canonical SMILESCC(C)(C)NCC(O)COc1ccc(NC(=O)NC2CCCCC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB11770
Drug NameTalinolol
CAS Number57460-41-0
Groups investigational
ATC Codes C07AB13
DescriptionTalinolol has been investigated for the basic science of Gastrointestinal Motility Disorder.

Categories: Adrenergic Agents Adrenergic Antagonists Adrenergic beta-Antagonists Agents causing hyperkalemia Alcohols Amines Amino Alcohols Antiarrhythmic agents Antihypertensive Agents Beta Blocking Agents, Selective Bradycardia-Causing Agents Cardiovascular Agents Cytochrome P-450 CYP2D6 Substrates Cytochrome P-450 Substrates Neurotransmitter Agents P-glycoprotein substrates Potential QTc-Prolonging Agents Propanols QTc Prolonging Agents
Cross-references: ChEBI: 135533 CHEMBL152067 ChemSpider: 62014 PubChem:68770 PubChem:347828123 RxCUI: 37546 Wikipedia: Talinolol
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08588 ADRB1 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P07550 ADRB2 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P10635 CYP2D6 Cytochrome P450 2D6 substrate enzymes
P08183 ABCB1 ATP-dependent translocase ABCB1 substrate transporters
Q92887 ABCC2 ATP-binding cassette sub-family C member 2 substrate transporters