Molecule Details
InChIKeyMVPXMHNFAQUXRM-UHFFFAOYSA-N
Compound Name2-(3-Chlorophenyl)-27-oxo-20-oxa-3,7,11,13-tetrazapentacyclo[19.3.1.13,6.115,19.09,13]heptacosa-1(25),9,11,15(26),16,18,21,23-octaene-18-carbonitrile
Canonical SMILESN#Cc1ccc2cc1Oc1cccc(c1)C(c1cccc(Cl)c1)N1CCC(NCc3cncn3C2)C1=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.6
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.6 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.1 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 6.1 IC50 ChEMBL