Molecule Details
InChIKeyMVLVSSYWLGSAFE-MAODMQOUSA-N
Compound Nametrans-(1R,2R)-N-(1-cyanocyclopropyl)-2-[(2R)-2-methyl-4-(3-methyl-1,2-benzoxazol-6-yl)piperazine-1-carbonyl]cyclohexane-1-carboxamide
Canonical SMILESCc1noc2cc(N3CCN(C(=O)[C@@H]4CCCC[C@H]4C(=O)NC4(C#N)CC4)[C@H](C)C3)ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43235 CTSK Homo sapiens Human PF08246 PF00112 7.8 IC50 ChEMBL;BindingDB
P07858 CTSB Homo sapiens Human PF00112 PF08127 6.2 IC50 ChEMBL;BindingDB
P25774 CTSS Homo sapiens Human PF08246 PF00112 6.1 IC50 ChEMBL;BindingDB