Molecule Details
InChIKeyMVJGBJOMTDVGRA-UHFFFAOYSA-N
Compound Name5-(3-(4-Methyl-sulfonylbenzene)-ureido)-[1,3,4]thiadiazole-2-sulfonic acid amide
Canonical SMILESCc1ccc(S(=O)(=O)NC(=O)Nc2nnc(S(N)(=O)=O)s2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.44
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00915 CA1 Homo sapiens Human PF00194 8.5 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 8.4 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.4 pIC50 TTD_MultiTarget