Molecule Details
InChIKeyMVCMGBIAYBTDLE-UHFFFAOYSA-N
Compound Name3-amino-6-(2-fluorophenyl)-N-(1-methyl-5-(piperidin-4-yloxy)-1H-pyrazol-4-yl)picolinamide
Canonical SMILESCn1ncc(NC(=O)c2nc(-c3ccccc3F)ccc2N)c1OC1CCNCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.4 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.3 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.6 Ki ChEMBL;BindingDB