Molecule Details
InChIKeyMUZRICFSRACWJI-UHFFFAOYSA-N
Compound Name[3-(3,4-Dichlorophenyl)-3-(3-spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylpropyl)piperidin-1-yl]-phenylmethanone
Canonical SMILESO=C(c1ccccc1)N1CCCC(CCCN2CCC3(CCc4ccccc43)CC2)(c2ccc(Cl)c(Cl)c2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 6.6 IC50 ChEMBL;BindingDB