Molecule Details
InChIKeyMUUSOYWTPTTZII-RMKNXTFCSA-N
Compound Name3-[4-((E)-3-Phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole
Canonical SMILESC(=C/c1ccccc1)\CN1CCN(CC2ON=C3c4ccccc4OCC32)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08913 ADRA2A Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P18825 ADRA2C Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB