Molecule Details
InChIKeyMUTUVLXBJKMVKT-RPBOFIJWSA-N
Canonical SMILESCC(=O)N1CCN(C(=O)N2C[C@H](c3ccc(F)cc3)[C@@H](N(C)C(=O)C(C)(C)c3cc(C(F)(F)F)cc(C(F)(F)F)c3)C2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25103 TACR1 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P29371 TACR3 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB