Molecule Details
InChIKeyMURRAGMMNAYLNA-UHFFFAOYSA-N
Compound NameImpromidine
Canonical SMILESCc1nc[nH]c1CSCCN=C(N)NCCCc1cnc[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.54
SourceBindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB20379
Drug NameImpromidine
CAS Number55273-05-7
Groups experimental
ATC Codes nan
DescriptionImpromidine is a small molecule drug. Impromidine has a monoisotopic molecular weight of 321.17 Da.

Categories: Amidines Guanidines Histamine Agents Histamine Agonists Imidazoles Neurotransmitter Agents
Cross-references: BindingDB: 50483127 CHEMBL12608 ZINC: ZINC000004216553
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H3N8 HRH4 Homo sapiens Human PF00001 7.9 Ki BindingDB
Q9Y5N1 HRH3 Homo sapiens Human PF00001 7.2 Ki BindingDB
DrugBank Target Actions (4)
Target Gene Target Name Action Type
P25021 HRH2 Histamine H2 receptor agonist targets
Q9H3N8 HRH4 Histamine H4 receptor agonist targets
Q9Y5N1 HRH3 Histamine H3 receptor agonist targets
P35367 HRH1 Histamine H1 receptor antagonist targets