Molecule Details
InChIKeyMUKGYZFIZLFCGL-LJQANCHMSA-N
Compound Name[(3R)-3-hydroxypyrrolidin-1-yl]-[3-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-2H-indazol-5-yl]methanone
Canonical SMILESCn1cc(-c2ccc(Cc3n[nH]c4ccc(C(=O)N5CC[C@@H](O)C5)cc34)cc2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 8.4 IC50 ChEMBL;BindingDB
Q9BWU1 CDK19 Homo sapiens Human PF00069 8.4 IC50 ChEMBL
P49336 CDK8 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB