Molecule Details
InChIKeyMUGOBVVTADQYDA-UHFFFAOYSA-N
Compound NameN-{2-[(4-cyanophenyl)[(1-methyl-1H-imidazol-5-yl)methyl]amino]ethyl}-1-methyl-N-[(4-phenylphenyl)methyl]-1H-imidazole-4-sulfonamide
Canonical SMILESCn1cnc(S(=O)(=O)N(CCN(Cc2cncn2C)c2ccc(C#N)cc2)Cc2ccc(-c3ccccc3)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.62
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5E175 rhlE Aliivibrio fischeri (strain ATCC 700601 / ES114) Pathogen PF00270 PF00271 6.6 IC50 BindingDB
Q5EI73 Plasmodium falciparum Pathogen PF01239 6.6 IC50 ChEMBL