Molecule Details
InChIKeyMTYMLJSBEPCLGC-ULIRXLGVSA-N
Compound Name(3R)-3-{[(2S)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl)acetyl]-oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Canonical SMILESO=C(O[C@H]1C[N+]2(CCCOc3ccccc3)CCC1CC2)[C@](O)(c1cccs1)C1CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08172 CHRM2 Homo sapiens Human PF00001 10.0 IC50 ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 9.9 IC50 ChEMBL;BindingDB
P20309 CHRM3 Homo sapiens Human PF00001 9.9 IC50 ChEMBL;BindingDB