Molecule Details
InChIKeyMTQBOVPCWAKWKD-UHFFFAOYSA-N
Compound Name1-Methyl-7-phenylmethoxy-6-pyridin-3-yl-3,4-dihydroquinolin-2-one
Canonical SMILESCN1C(=O)CCc2cc(-c3cccnc3)c(OCc3ccccc3)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11511 CYP19A1 Homo sapiens Human PF00067 8.0 IC50 ChEMBL;BindingDB
P15538 CYP11B1 Homo sapiens Human PF00067 6.9 IC50 ChEMBL;BindingDB
P19099 CYP11B2 Homo sapiens Human PF00067 6.8 IC50 ChEMBL;BindingDB