Molecule Details
InChIKeyMTMZZIPTQITGCY-OLGWUGKESA-N
Canonical SMILESC#C[C@]1(O)CC[C@H]2[C@@H]3CCc4cc(O)ccc4[C@H]3[C@@H](OC)C[C@@]21C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB13418
Drug NameMoxestrol
CAS Number34816-55-2
Groups experimental
ATC Codes G03CB04
Descriptionnan

Categories: Estradiol Congeners Estrogen Antagonists Estrogenic Steroids, Alkylated Estrogens Fused-Ring Compounds Genito Urinary System and Sex Hormones Gonadal Hormones Gonadal Steroid Hormones Hormone Antagonists Hormones Hormones, Hormone Substitutes, and Hormone Antagonists Norpregnanes Norpregnatrienes Norsteroids Sex Hormones and Modulators of the Genital System Steroids Synthetic Estrogens, Plain
Cross-references: BindingDB: 50218560 ChEBI: 34857 CHEMBL1628161 ChemSpider: 10128336 C14757 Wikipedia: Moxestrol ZINC: ZINC000003815417
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P03372 ESR1 Homo sapiens Human PF12743 PF00104 PF02159 PF00105 8.6 IC50 ChEMBL;BindingDB
Q92731 ESR2 Homo sapiens Human PF12497 PF00104 PF00105 8.6 IC50 ChEMBL