Molecule Details
InChIKeyMTEAPQJRNVJOCS-UHFFFAOYSA-N
Compound Name3-Hydroxy-3-phenyl-2-({[(4-sulfamoylphenyl)amino]thioxomethyl}amino)propanoic acid
Canonical SMILESNS(=O)(=O)c1ccc(N/C(S)=N/C(C(=O)O)C(O)c2ccccc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.34
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.7 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.7 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.6 Ki ChEMBL;BindingDB