Molecule Details
InChIKeyMSOZBJDLTCXBAV-JOCHJYFZSA-N
Compound NamePyrimidylpyrrole, 11d
Canonical SMILESCc1cc(Cl)ccc1Nc1ncc(C)c(-c2c[nH]c(C(=O)N[C@H](CO)c3cccc(Cl)c3)c2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 8.3 Ki ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.1 pIC50 TTD_MultiTarget
O14965 AURKA Homo sapiens Human PF00069 6.4 Ki ChEMBL;BindingDB