Molecule Details
InChIKeyMSDVVDOJAWEWIF-NASUQTAISA-N
Canonical SMILESCOc1nc(-c2cccc(-c3cccc(-c4ccc(C(C)N5CC6(CN(C(C)=O)C6)C5)c(OC)n4)c3Cl)c2Cl)ccc1CNC[C@@H]1CCC(=O)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NZQ7 CD274 Homo sapiens Human PF08205 PF07686 6.5 IC50 ChEMBL
Q9BQ51 PDCD1LG2 Homo sapiens Human PF22705 6.4 IC50 ChEMBL;BindingDB